Abstract
2,6-Diamino-4,N-diarylpyridines were identified as potent, isoform selective inhibitors of the enzymatic activity of lysophosphatidic acid acyltransferase-beta (LPAAT-beta).
MeSH terms
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Acyltransferases / antagonists & inhibitors*
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Enzyme Inhibitors / chemical synthesis*
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Enzyme Inhibitors / pharmacology
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Humans
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Inhibitory Concentration 50
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Isomerism
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Protein Isoforms
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Pyridines / chemical synthesis*
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Pyridines / pharmacology
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Structure-Activity Relationship
Substances
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Enzyme Inhibitors
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Protein Isoforms
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Pyridines
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Acyltransferases
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2-acylglycerophosphate acyltransferase